What are the indications for and evidence behind the use of tamsulosin and finasteride in women?

Comment by InpharmD Researcher

Numerous trials have investigated the use of tamsulosin and finasteride in women. Tamsulosin has been used off-label in women for the treatment of lower urinary tract symptoms (LUTS), including urinary frequency/urgency, decreased force of stream, hesitancy, need to strain, feeling of incomplete bladder emptying, and ureteral stones. Significant improvement with tamsulosin has been demonstrated over placebo for many LUTS-related outcomes, including International Prostate Symptom Score (IPSS), quality-of-life (QoL) score, and Overactive Bladder Questionnaire (OAB-q). The most notable off-label use of finasteride in women is for hair loss, as well as hirsutism and alopecia, with some clinical studies demonstrating favorable outcomes. However, other literature determined a lack of conclusive data regarding its effectiveness. Many relevant studies are limited due to relatively small sample sizes.

Background

A 2017 systematic review and meta-analysis evaluated the efficacy and safety of tamsulosin for the treatment of lower urinary tract symptoms (LUTS) in women. A total of 6 randomized controlled trials (RCTs) were included (N= 764 female patients). International Prostate Symptom Score (IPSS), quality-of-life (QoL) score, and Overactive Bladder Questionnaire (OAB-q) were among the scales used to compare outcomes. Total IPSS improvement was evaluated in two RCTs. Compared to placebo, tamsulosin was found to be significantly more effective in improving total IPSS, with a pooled estimate of standardized mean difference (SMD) of -4.08 (95% confidence interval [CI] -5.93 to -2.23, p<0.00001). For the IPSS storage symptom score, two RCTs again demonstrated the superiority of tamsulosin compared to placebo, with an SMD of -3.16 (95% CI -4.47 to -1.85). Both of these comparisons included significant heterogeneity (I2= 57%, p= 0.13 and I2= 94%, p<0.0001, respectively). Only one RCT included IPSS voiding symptom score, finding improvement with tamsulosin when compared to placebo, with a MD of -2.40 (95% CI -3.71 to -1.09). No significant differences were demonstrated when comparing tamsulosin vs. solifenacin or tolterodine combined with tamsulosin for any IPSS scores. [1]

For QoL score, two RCTs demonstrated the superiority of tamsulosin compared to placebo, with a pooled estimate of SMD of -2.1 (95% CI -2.67 to -1.71), again with significant heterogeneity (I2= 84%, p= 0.01). Similar to previous comparisons, no significant difference was revealed between tamsulosin compared to solifenacin or tolterodine combined with tamsulosin. Only one included RCT evaluated OAB-q, finding a significant improvement in QAB-q with tamsulosin compared to placebo (MD -5.60 [95% CI -6.59 to -4.61]), but not between tamsulosin and solifenacin. Results from a voiding diary were evaluated in one RCT, demonstrating significant improvement in voiding volume with tamsulosin vs. placebo (MD -7.50 [95% CI -10.26 to -4.74]), but with no difference for the daily number of voids, incontinence episodes per day, urgency episodes, and nocturia episodes between the two groups. Significant improvement with tamsulosin was found in some urodynamic parameters as evaluated in 3 RCTs. Compared to prazosin, tamsulosin was found to boost average flow rate (MD -1.78 [95% CI -3.32 to -0.24]), and compared to tamsulosin combined with tolterodine, tamsulosin alone was found to improve post-void residual volume (PVR; MD 24.30 [95% CI 16.34 to 32.26]). The presented data suggest tamsulosin to be an effective treatment option for LUTS in women, however, larger, adequately-powered RCTs are still required to further solidify its efficacy. [1]

A 2018 systematic review focused on the safety of tamsulosin in women and children. Ultimately, 49 studies were found including a mix of men and women, 4 studies with only women, and 3 studies with children. Cumulatively, 725 women and 290 children were included. In studies specific to women participants (age 18 to 70 years, treated for LUTS or overactive bladder), adverse events reported included headache, orthostatic hypotension, incontinence, lethargy, dizziness, drowsiness, asthenia, dry mouth, constipation, nausea, abdominal pain, and dyspepsia; no serious adverse events were reported in these studies. In pediatric studies (mean age range 7.3 to 8.2 years, treated for neuropathic bladder or ureteral stones), nasal congestion, somnolence, and headache were reported. One pediatric death was also reported, considered potentially related to the study drug. In general, the most common adverse events documented in this review, including in women and children, were consistent with known adverse events of tamsulosin reported among men with LUTS secondary to benign prostatic hyperplasia. [2]

A 2019 systematic review evaluated the efficacy and use of finasteride in women with a focus on dosage, length of treatment, and conditions that can benefit from finasteride therapy. A total of 65 studies (published RCTs, prospective cohort studies, retrospective studies, and case reports) involving 2,683 patients were included in the final analysis. The majority of the female patients included in the studies were treated with finasteride for hirsutism (48.7%). The efficacy of finasteride use on female pattern hair loss (FPHL) was assessed in 34.7% of RCTs; while other forms of hair loss such as alopecia, lichen planopilaris, and frontal fibrosing alopecia were studied, no RCTs that evaluated finasteride therapy for those conditions were identified. The analysis of other prospective and retrospective studies demonstrated that finasteride may improve hair loss in women with FPHL or frontal fibrosing alopecia. Evidence from RCTs suggested that finasteride treatment can improve hirsutism scores in women with hirsutism or idiopathic hirsutism secondary to polycystic ovarian syndrome. In general, the doses of oral finasteride ranged from 0.5 to 5 mg/day in females between the age of 6 to 88 years with the length of treatment ranging from 6 to 12 months (57.6%). Monotherapy was used in 88.9% of included finasteride patients and a continuous frequency of use was implemented in 96.4% of finasteride patients. Several recommendations regarding finasteride use in women along with the corresponding references were made by the authors and are summarized in Table 5. [3]

A 2015 Cochrane systematic review investigated interventions for hirsutism in women with polycystic ovary syndrome, idiopathic hirsutism, or idiopathic hyperandrogenism. Two included studies suggested a difference in reduction of Ferriman‐Gallwey hirsutism assessment scores for finasteride 5 mg to 7.5 mg daily compared to placebo (MD ‐5.73, 95% CI ‐6.87 to ‐4.58), however, the authors determined this very low quality of evidence was unlikely to be clinically meaningful. Two studies were also included comparing finasteride vs. spironolactone, finding similar effectiveness (MD 1.49, 95% CI ‐0.58 to 3.56 vs. MD 0.40, 95% CI ‐1.18 to 1.98). This was also considered to be low-quality data, and ultimately the authors determined that finasteride showed inconsistent results, precluding any firm conclusions. [4]

Another 2018 systematic review and meta-analysis compared pharmacologic treatments for hirsutism in women. A total of 43 RCTs were analyzed and six drug classes or combination of classes were used, including oral contraceptive pills (OCPs), antiandrogen, insulin sensitizer, OCPs plus antiandrogen, OCPs plus insulin sensitizer, and antiandrogen plus insulin sensitizer. When compared with placebo, antiandrogen monotherapy with finasteride presented with a significant reduction in hirsutism with an overall effect size of −1.48 (95% CI −2.18 to −0.78, p<0.05). While antiandrogen monotherapy with flutamide, finasteride, and spironolactone was demonstrated to be more effective than placebo, all these agents had similar efficacy when compared to each other. A combination of OCPs with finasteride demonstrated superior efficacy in comparison with placebo with an effect size of −1.64 (95% CI −2.72 to −0.55). It should be noted that the risk of bias in the included trials was high. Furthermore, as many of the studies had important methodological limitations, the precision of the results remains limited, and the interpretation of data should be done with caution. [5]

References:

[1] Zhang HL, Huang ZG, Qiu Y, Cheng X, Zou XQ, Liu TT. Tamsulosin for treatment of lower urinary tract symptoms in women: a systematic review and meta-analysis. Int J Impot Res. 2017;29(4):148-156. doi:10.1038/ijir.2017.12
[2] Kaplan SA, Chughtai BI. Safety of Tamsulosin: A Systematic Review of Randomized Trials with a Focus on Women and Children. Drug Saf. 2018;41(9):835-842. doi:10.1007/s40264-018-0674-y
[3] Hu AC, Chapman LW, Mesinkovska NA. The efficacy and use of finasteride in women: a systematic review. Int J Dermatol. 2019;58(7):759-776. doi:10.1111/ijd.14370
[4] van Zuuren EJ, Fedorowicz Z, Carter B, Pandis N. Interventions for hirsutism (excluding laser and photoepilation therapy alone). Cochrane Database Syst Rev. 2015;2015(4):CD010334. Published 2015 Apr 28. doi:10.1002/14651858.CD010334.pub2
[5] Barrionuevo P, Nabhan M, Altayar O, et al. Treatment Options for Hirsutism: A Systematic Review and Network Meta-Analysis. J Clin Endocrinol Metab. 2018;103(4):1258-1264. doi:10.1210/jc.2017-02052

Literature Review

A search of the published medical literature revealed 7 studies investigating the researchable question:

What are the indications for and evidence behind the use of Tamsulosin and finasteride in women?

Level of evidence

B - One high-quality study or multiple studies with limitations  Read more→



Please see Tables 1-7 for your response.


The Effectiveness of Tamsulosin in Treating Women With Voiding Difficulty

Design

Prospective study

N=97

Objective

To evaluate the effectiveness of tamsulosin monotherapy in treating women with chronic voiding difficulty

Study Groups

Bladder outlet obstruction (n=33)

Detrusor underactivity (n=52)

Equivocal (n=12)

Inclusion Criteria

Female patients visiting a neurological clinic with the predominant complaint of chronic, bothersome voiding symptoms; accepted tamsulosin treatment

Exclusion Criteria

Mechanical obstruction, indwelling catheterization, self-intermittent catheterization, concurrent use of medications that may affect voiding

Methods

Patients were treated with 0.2 tamsulosin daily for 6 or more weeks. Doses were not increased during the 6-week study period.  Patients were returned at week 2 for evaluation of adverse events and at week 6 for evaluation of therapeutic outcome.

Patients were asked to compare the current voiding condition to baseline using a 5-point scale: 0, worsened: 1, little of no change (<25% improvement); 2, slightly improved (25-50%), 3, moderately improved (50-75%); 4, markedly improved (75% or greater).

Duration

Treatment: 6 weeks

Outcome Measures

Subjective: global assessment and self-administered Internation Prostate Symptoms Score (IPSS) questionnaire

Objective: maximum flow rate (Qmax), post-void residual urine (PVR), voiding efficiency

Baseline Characteristics

 

All patients (n=97)

   

Age, years (range)

63.8 ± 12.9 (19-87)    

Comorbidities leading to voiding difficulty

Diabetes

History of pelvic operation including hysterectomy

Parkinson

Colorectal operation

Herniation

 

20 (21%)

14 (14%)

5 (5%)

3 (3%)

3 (3%)

   

Results

 

Baseline

Endpoint

P-value
Total IPSS score

20.2 ± 7.2

14.8 ± 7.4 <0.01

Voiding symptom score

Abdominal straining

Intermittency

Weak stream

Incomplete emptying

12.9  5.2

3.0 ± 1.9

3.5 ± 1.7

3.1 ± 1.7

3.3 ± 1.8

8.6 ± 6.2

2.2 ± 1.9

2.2 ± 2.1

2.1 ± 1.9

2.1 ± 2.1

<0.01

<0.01

<0.01

<0.01

<0.01

Storage symptom score

Frequency

7.3 ± 3.7

2.9 ± 1.7

6.2 ± 3.4

2.3 ± 1.9

<0.01

<0.01

Qmax, mL/s

10.4  3.4

14.1  6.3

<0.01

Post-void residual urine, mL

123.1 ± 108.8

71.1 ± 73.3 <0.01
Voiding efficiency, %

64.2 ± 24.1

77.3 ± 18.0 <0.01

There were no significant differences in the change from baseline in storage symptom scores of urgency and nocturia at the end of the study.

A subgroup analysis was performed to compare the effect of tamsulosin in 85 patients classified as bladder outlet obstruction (n=33) and detrusor underactivity (n=52). Improvements for total IPSS, Qmax, PVR, and voiding efficiency were similar between both groups, but those with bladder outlet obstruction had a more favorable reduction in voiding symptom score compared to those with detrusor underactivity (P=0.03).

Adverse Events

Dizziness (7.1%), skin itching (5.1%), asthenia (4.1%), rhinitis (4.1%), stress incontinence (3.1%), ankle edema (1.0%)

Study Author Conclusions

Although hampered by the fact that it was not being placebo‐controlled, this study suggests that tamsulosin improves voiding symptoms and urodynamic parameters in nearly one‐third of women with voiding difficulty and comparable good therapeutic response rates were observed between patients with bladder outlet obstruction and detrusor underactivity.

InpharmD Researcher Critique

This study was not placebo-controlled not randomized due to its small population size. This study only included patients who accepted tamsulosin treatment, which may contribute to selection bias of optimal patients. The patients all had different characteristics that contributed to their voiding difficulty. Because a lower dose of tamsulosin was used, it was not known if patients were underdosed. 

References:

Chang SJ, Chiang IN, Yu HJ. The effectiveness of tamsulosin in treating women with voiding difficulty. Int J Urol. 2008;15(11):981-985. doi:10.1111/j.1442-2042.2008.02134.x

α1-Blockers For The Treatment Of Recurrent Urinary Tract Infections In Women With Dysfunctional Voiding: A Prospective Randomized Study

Design

Prospective, open-label, multicenter, randomized study

N=128

Objective

To evaluate the therapeutic effects of tamsulosin on recurrent urinary tract infections (UTIs) in women with dysfunctional voiding

Study Groups

Uroflowmetry biofeedback (n=35)

Tamsulosin (n=38)

Uroflowmetry biofeedback plus tamsulosin (n=37)

No treatment (n=18)

Inclusion Criteria

Women with recurrent UTI and dysfunctional voiding

Exclusion Criteria

Patients with anatomical abnormalities

Methods

Women with recurrent urinary tract infections and dysfunctional voiding were included and randomly assigned to the following groups: uroflowmetry biofeedback; tamsulosin 0.4 mg once daily; uroflowmetry biofeedback combined with tamsulosin 0.4 mg once daily; and no treatment. Patients were evaluated by the American Urological Association Symptom Index at 3, 6, and 12 months.

At the beginning of the study, biofeedback training was carried out weekly for 10 weeks. After the patients understood the concept, sessions were scheduled at 4-week intervals and continued for 12 months. Tamsulosin was given for 3 months, then stopped.

Duration

Follow-up: 1 year 

Outcome Measures

Storage symptoms (frequency and urgency)

Emptying symptoms (decreased force of stream, hesitancy, need to strain and a feeling of incomplete bladder emptying)

Baseline Characteristics

  Uroflowmetry biofeedback (n=35)

Tamsulosin (n=38)

Uroflowmetry biofeedback plus tamsulosin (n=37) No treatment (n=18)

Storage symptoms 

27 (77.1%) 27 (71%)  29 (78.4%) 11 (61.1%)

Emptying symptoms

27 (77.1%) 24 (63.1%) 25 (65.7%) 11 (61.1%) 

Voiding volume, mL

397 ± 45 389 ± 88 395 ± 85 387.2 ± 50

The mean age of participants was 25.3 years (range, 18-34)

Results

 

Uroflowmetry biofeedback (n=35)

Tamsulosin (n=38)

Uroflowmetry biofeedback plus tamsulosin (n=37)

No treatment (n=18)

Storage symptoms 

3 months

6 months

1 year

 

18 (51.4%)

15 (55.5%)

16 (59.2%)

 

25 (65.7%)

18(60%) 

20 (66.6%)

 

15 (40.5%)

12 (42.8%)

11 (39.2)

 

11 (61.1%)

11( 61.1%)

11 (61.1)

Emptying symptoms

3 months

6 months

1 year

 

20 (57.1%)

16 (59.2%)

15 (55.5%)

 

21 (55.2%)

18(60%) 

19 (63.3%)

 

15 (40.5%)

10 (35.7%)

11 (39.2)

 

11 (61.1%) 

11 (61.1%) 

11 (61.1%) 

Voiding volume, mL

3 months

6 months

1 year

 

473 ± 44

472 ± 48

460 ± 37

 

459 ± 70

458 ± 49

462 ± 55

 

492 ± 58

498 ± 49

469 ± 50

 

N/A

N/A

377 ± 3.3

By the analysis of the urodynamic parameters, the mean opening detrusor pressure and detrusor pressure at maximum flow decreased significantly after treatment in all three groups (with a better outcome in patients of group 3; P<0.05) and remained stable during the follow-up period.

The prevalence of UTI decreased significantly in all groups after treatment (P<0.05), and the results remained stable in the follow-up period

Adverse Events

No adverse effects were recorded in the patients during the treatment with each modality

Study Author Conclusions

In women with dysfunctional voiding and recurrent urinary tract infection, tamsulosin associated with uroflowmetry biofeedback might be an effective and safe treatment option for improving urinary symptoms and quality of life.

InpharmD Researcher Critique

This study is limited by its relatively small sample size and single-center design. Baseline characteristics of participants were not reported. The results of this study may be affected by the Hawthorne effect, a bias that exists when subjects know they are being observed. Since patients were aware of their voiding frequency, liquid intake being adjusted, and measuring voided volume, some participants may have made lifestyle adjustments to supplement the potential effects of their treatments. Pelvic floor therapy may also have an indirect effect on storage symptoms.

References:

Minardi D, Pellegrinelli F, Conti A, et al. α1-Blockers for the treatment of recurrent urinary tract infections in women with dysfunctional voiding: a prospective randomized study. Int J Urol. 2015;22(1):115-121. doi:10.1111/iju.12601

Efficacy and safety of tamsulosin in medical expulsive therapy for distal ureteral stones with renal colic: a multicenter, randomized, double-blind, placebo-controlled trial

Design

Multicenter, randomized, double-blind, placebo-controlled trial

N=3,296

Objective

To evaluate the efficacy and safety of tamsulosin for distal ureteral stones compared with placebo

Study Groups

Tamsulosin (n=1,642)

Placebo (n=1,654)

Inclusion criteria

Age 18 to 60 years old, emergency admission for renal colic, the presence of single uteral stone, stone in the distal ureter (4 to 7 mm), unilateral presentation

Exclusion criteria

Fever, urinary tract infection, severe hydronephrosis, renal insufficiency (GFR < 60 mL/min), abnormal anatomy, history of ureter strictures, diabetes mellitus, hypotension (systolic blood pressure <100 mm Hg), known or suspected pregnancy, current use of alpha-adrenoceptor antagonists or corticosteroids, previous history of ipsilateral ureteral surgery, spontaneous stone expulsion, known or suspected allergy to the study medications

Methods

 

Patients were randomized (1:1) to receive either two capsules of tamsulosin 0.2 mg or placebo. Medication or placebo was taken for up to four weeks or until spontaneous stone passage.

Duration

September 2011 and August 2013

Four-week treatment period

Outcome Measures

Stone expulsion rate, average time to expulsion, rate of pain relief therapy during treatment period, side effects

Baseline Characteristics

 

Tamsulosin (n=1,642)

Placebo (n=1,654)

 

Age, years

40.1 40.7  

Women

556 (34%) 605 (37%)  

Stone size, mm

5.8 5.7  

Stone size < 5 mm

555 (34%) 561 (34%)  

Stone size > 5 mm

1,087 (66%) 1,093 (66%)  

Results

 

Tamsulosin (n=1,642)

Placebo (n=1,654)

p-value

Stone expulsion rate, No.

1,419 (86%) 1,300 (79%) <0.001

Average stone expulsion time, hour

148.3 248.7 <0.001

Rate of pain relief therapy

31 (1.9%) 155 (9.4%) <0.001

Side effect

92 (5.6%) 84 (5.1%) <0.001

Adverse Events

Tamsulosin: dizziness (3.2%), headache (2.5%), nausea (2.6%), vomiting (2.3%), retrograde ejaculation (6.2%)

There was no significant difference in adverse effects compared to the placebo group

Study Author Conclusions

The use of tamsulosin significantly facilitates the passage of distal ureteral stones and relieves renal colic.

InpharmD Researcher Critique

A strength of this study is that it was randomized, double-blinded, and placebo-controlled, which therefore reduces the amount of bias that can be introduced into the results. However, the exclusion criteria was extensive which may have introduced a biased patient selection.

References:

Ye Z, Zeng G, Yang H, Tang K, Zhang X, Li H, et al. Efficacy and safety of tamsulosin in medical expulsive therapy for distal ureteral stones with renal colic: A multicenter, randomized, double-blind, placebo-controlled trial. Eur Urol. 2017: S0302-2838(17)30972-7.

Effect of Tamsulosin on Passage of Symptomatic Ureteral Stones

Design

Randomzied, double-blind, placebo-controlled trial

N=512

Objective

To determine if tamsulosin promotes the passage of urinary stones within 28 days among emergency department patients

Study Groups

Tamsulosin (n=267)

Placebo (n=245)

Inclusion Criteria

18 years olds or older presenting to the emergency room with symptomatic urinary store determined by computed tomography (CT) to be less then 9 mm in diameter and located in the ureter

Exclusion Criteria

None reported

Methods

Participants were randomized 1:1 to either tamsulosin 0.4 mg or matching placebo once daily for 28 days.

Study participants were contacted by telephone to collect data at 2, 7, 15, 20, 29, and 90 days after randomization. Study participants enrolled in the second phase were also asked to undergo a follow-up CT scan after the 28-day treatment period to determine whether their stone had passed based on this imaging modality.

Duration

Treatment: 28 days

Follow-up: 90 days

Outcome Measures

Primary: the passage of ureteral stone within 28 days

Secondary: participants who discontinued their assigned study medication and crossed over to open-label tamsulosin; safety

Baseline Characteristics

 

Tamsulosin (n=267)

Placebo (n=245) 

Age, years

41.8 ± 13.6 39.3 ± 12.9

Female

70 (26.2%) 69 (28.2%)

Past history of kidney stone

76 (28.5%) 76 (31%)

Symptomatic stone size on CT, mm

3.8 ± 1.4 3.7 ± 1.4

Results

 

Tamsulosin (n=267)

Placebo (n=245)

P-value

Patient-reported stone passage

128/258 (49.6%) 113/245 (47.3%) 0.60

Stone passed on follow-up CT

 

102/122 (83.6%)

90/116 (77.6%)

 

0.24

Crossover to open-label tamsulosin

15/214 (7.0%)

14/189 (7.4%)

0.88

Adverse Events

Common Adverse Events: upset stomach, nausea, or vomiting,(24% vs 25%); abdominal pain or stomach ulcer (15% vs 19%); dizziness (12% vs 9%); tachycardia (1.9% vs 3.7%); urinary tract infections (1.4% vs 2.1%)

No serious adverse events were reported.

Study Author Conclusions

Tamsulosin did not significantly increase the stone passage rate compared with placebo. These findings do not support the use of tamsulosin for symptomatic urinary stones smaller than 9 mm. Guidelines for medical expulsive therapy for urinary stones may need to be revised.

InpharmD Researcher Critique

Unlike previous clinical trials, this trial had limited enrollment of patients with distal ureteral stones. Other limitations of the study include the potential lack of generalizability of our findings to patients seen outside of a US tertiary care center that allows for easy access to urologists and high rates of surgery for larger stones. In addition, a high proportion of our participants had stones smaller than 5 mm in diameter.

This study also did not assess for urologic parameters, such as increased urine output.

References:

Meltzer AC, Burrows PK, Wolfson AB, et al. Effect of Tamsulosin on Passage of Symptomatic Ureteral Stones: A Randomized Clinical Trial. JAMA Intern Med. 2018;178(8):1051-1057. doi:10.1001/jamainternmed.2018.2259

Summary of recommendations for finasteride treatment in women
Recommendation Grade of recommendation Quality of evidence Source
Finasteride can be used to treat females with IH or hirsutism secondary to PCOS 1 A Faloia et al.; Petrone et al.; Bayram et al.; Bayram et al.; Lakryc et al.; Tartagni et al.; Tartagni et al.
Topical finasteride can be used to treat women with IH 1 A Lucas; Tahvilian et al.; Alijanpour
For shorter courses of treatment, finasteride is more effective than flutamide in treating females with IH or hirsutism secondary to PCOS 1 A Falsetti et al.
Medium-dose finasteride (2.5 mg/day) is just as effective as high-dose finasteride (5 mg/day) for treating females with IH or hirsutism secondary to PCOS 1 A Bayram et al.
Finasteride is just as effective as flutamide, spironolactone, and CPA+EE for treating females with IH or hirsutism secondary to PCOS 1 A Fruzzetti et al.; Moghetti et al.; Beigi et al.
Finasteride is less effective than flutamide, spironolactone, CPA+EE, and GnRH in treating females with IH or hirsutism secondary to PCOS 1 A Erenus et al.; Sahin et al.; Falsetti
et al.; Venturoli et al.; Bayhan et al.; Muderris et al.; Lumachi et al
Combination therapy of finasteride and spironolactone or finasteride and CPA+EE is more effective than monotherapy in treating IH or hirsutism secondary to PCOS 1 A Tartagni et al.; Sahin et al.; Unluhizarci et al.; Kelestimur et al.
Combination therapy of finasteride and rFSH can be used to treat females with PCOS 1 A Tartagni et al.
Finasteride does not alter the volume and number of cysts in female ovaries 1 A Arie et al.
Finasteride is less effective than flutamide and CPA+EE in treating females with acne 1 A Carmina and Lobo
AR-CAG repeat numbers can predict finasteride efficacy in Caucasian females with FPHL 1 A Keene et al. 
Lower-dose finasteride (1 mg/day) and high-dose finasteride (5 mg/day) are not effective for treating hair loss in females with FPHL 1 A Whiting et al.; Price and Roberts et al.; Altomare et al.; Carmina and Lobo
Topical finasteride is not effective for treating hirsutism 2A A Price and Allen et al.
Combination therapy of finasteride and flutamide is more effective than monotherapy in treating hirsutism 2A B Unluhizarci et al.
Finasteride can improve symptoms in females with acne and alopecia 2A B Kohler et al.
AR-CAG repeat numbers cannot predict finasteride efficacy in Japanese females with FPHL 2A B Yamazaki et al.
Low to high-dose finasteride (1.25–5 mg/day) can improve hair loss in females with FPHL 2A B Shum et al.; Thai et al.; Yeon et al.; Boychenko et al.; Oliveira-Soares et al.; Boersma et al.
Low-dose finasteride (1.25 mg/day) or combination therapy of finasteride and minoxidil is not effective for treating hair loss in females with FFA 2A B Rallis et al.; Kim et al.
Finasteride can improve hair loss in females with FFA 2A B Tosti et al.; Ladizinski et al.; Vano-Galvan et al.
Finasteride therapy does not alter follicular development or ovulation 2A B Wong et al.
Finasteride can cause mood disturbances in females with FPHL 2B B Altomare et al.
Finasteride can improve hair loss in female-to-male transgender patients with FPHL 2B B Moreno-Arrones et al.
Combination therapy of finasteride, cetirizine, and a topical medication can mildly improve symptoms of CLPP and FFA 2B B Mardones et al.
Finasteride can resolve SRF in females with central serous chorioretinopathy 2B B Moisseiev et al.
Combination therapy of finasteride, minoxidil, and triamcinolone acetonide can improve hair loss in females with FFA 2B C Moreno-Ramirez et al. 
Finasteride can improve symptoms in females with HS 2B C Farrell et al.; Joseph et al.; Khandalavala; Mota et al.
Finasteride can be used to alleviate chronic migraines in females 2B C Check et al.
Finasteride cessation can stop seizures in females 2B C Pugnaghi et al.
Finasteride therapy prior to pregnancy can result in successful full-term pregnancy and live birth 2B C Tartagni et al.
Unintentional finasteride during early pregnancy can cause aphalangia in a newborn girl 2B C Sallout and Alwadi

According to criteria by Robinson et al: Grade of recommendation: 1, strong recommendation; high-quality, patient-oriented evidence; 2A, weak recommendation; limited-quality, patient-oriented evidence; 2B, weak recommendation; low-quality evidence. Quality of evidence: A, systematic review/meta-analysis; randomized clinical trials with consistent findings; all-or-none observational studies; B, systematic review/ meta-analysis of lower-quality clinical trials or studies with limitations and inconsistent findings; lower-quality clinical trial; cohort study; case-control study; C, consensus guidelines, usual practice, expert opinion, case series.

AGA, androgenetic alopecia; AR-CAG, androgen receptor cytosine, adenine, guanine; CLPP, classic lichen planopilaris; CPA, cyproterone acetate; CSCR, central serous chorioretinopathy; EE, ethinyl estradiol; FAGA, female androgenic alopecia; FFA, frontal fibrosing alopecia; FPHL, female pattern hair loss; HS, hidradenitis suppurativa; IH, idiopathic hirsutism; PCOS, polycystic ovary syndrome; SRF, subretinal fluid.

References:

Adapted from:
Hu AC, Chapman LW, Mesinkovska NA. The efficacy and use of finasteride in women: a systematic review. Int J Dermatol. 2019;58(7):759-776. doi:10.1111/ijd.14370

The effectiveness of finasteride and dutasteride used for 3 years in women with andorgenetic alopecia

Design

Retrospective cohort study

N=120

Objective

To evaluate the effectiveness of finasteride and dutasteride on hair loss in women with androgenetic alopecia over a period of 3 years

Study Groups

Finasteride (n=60)

Dutasteride (n=60)

Inclusion criteria

Clinical diagnosis of Ludwig grade 1 or grade 2 androgenetic alopecia confirmed by the presence of thin hair on a microscopic picture, continuous treatment for at least 3 years (assessed by regular filling of the prescription)

Exclusion criteria

N/A

Methods

Patients received either finasteride 1.25 mg daily or dutasteride 0.15 mg daily. An increase in hair thickness was obtained by subtracting the pretreatment hair thickness from that measured after 3 years. Treatment was considered effective if the hair thickness increase was equal to, or greater than zero. 

Duration

10 years

Outcome Measures

Hair thickness

Baseline Characteristics

 

Finasteride (n=60)

Dutasteride (n=60)

 

Age, years

   < 50

   > 50

 

30 (50%)

30 (50%)

 

30 (50%)

30 (50%)

Results

 

HTI<0 mm

HTI≥0 mm

Effectiveness

Finasteride 1.25 mg

   <50 years

   ≥50 years

   All ages

 

5

6

11

 

25

24

49

 

83.3%

80%

81.7%

Dutasteride 0.15 mg

   <50 years

   ≥50 years

   All ages

 

5

5

10

 

25

25

50

 

83.3%

83.3%

83.3%

Overall

21

99

82.5%

HTI=hair thickness increase

All hair thickness increases were statistically significantly different from 0 in both age categories and at all sites of the scalp (P<0.05), except for the increase in the age category above 50 years by dutasteride at the frontal site.

Dutasteride had higher means for users in the age group under 50 at the center of the scalp and the vertex (P<0.05).

Adverse Events

Not disclosed

Study Author Conclusions

Finasteride 1.25 mg and dutasteride 0.15 mg given daily for 3 years effectively increased hair thickness and arrested further deterioration in women with androgenetic alopecia.

InpharmD Researcher Critique

The study provides evidence that dutasteride may be better than finasteride for increasing hair thickness in women with alopecia but there was no control or double-blind data and more studies are needed for conclusive evidence. Additionally, only hair thickness was measured instead of growth density.

References:

Boersma IH, Oranje AP, Grimalt R, Iorizzo M, Piraccini BM, Verdonschot EH. The effectiveness of finasteride and dutasteride used for 3 years in women with androgenetic alopecia. Indian J Dermatol Venereol Leprol. 2014;80(6):521-5.

Clinical and endocrine effects of finasteride, a 5 alpha-reductase inhibitor, in women with idiopathic hirsutism

Design

Randomized, single-blind study

N=18

Objective

To evaluate the effects of long-term administration of finasteride on hirsutism score, basal gonadotropin and androgen secretion in women with idiopathic hirsutism

Study Groups

Finasteride (n=9)

Placebo (n=9)

Inclusion criteria

Women with moderate to severe hirsutism 

Exclusion criteria

Acne-seborrhea, clinical signs of hyperandrogenism

Methods

Patients were randomized to receive finasteride 7.5 mg or placebo daily for 9 months.

Duration

9 months

Outcome Measures

Reduction in hirsutism score, biomarker levels

Baseline Characteristics

 

Finasteride (n=9)

Placebo (n=9)

Age, years

20.9 ± 0.62 20.2 ± 0.62

Ferriman-Gallway score

21.8 ± 0.81 19.0 ± 1.57

Results

 

Placebo (n=9)

Finasteride (n=9)

Unbound testosterone, pg/mL

Baseline

3 months

6 months

9 months

 

2.7 ± 0.08

2.88 ± 0.14

2.82 ± 0.1

2.92 ± 0.09

 

2.97 ± 0.13

2.90 ± 0.13

2.97 ± 0.11

3.04 ± 0.08

The Ferriman and Gallwey hirsutism score of patients treated with finasteride was statistically significant when compared to placebo (p<0.05), but there was no significant change in the placebo group.

Adverse Events

Not disclosed

Study Author Conclusions

Finasteride decreased the hirsutism score of patients affected by idiopathic hirsutism with few sides during treatment.

InpharmD Researcher Critique

A limitation of the study is the small sample size. This study did not report individual Ferriman and Gallwey hirsutism scores other than the baseline.

 
References:

Ciotta L, Cianci A, Calogero AE, et al. Clinical and endocrine effects of finasteride, a 5 alpha-reductase inhibitor, in women with idiopathic hirsutism. Fertil Steril. 1995;64(2):299-306.