Is it safe to use TXA perioperatively in a patient who has a history of stroke, DVT, and sickle cell disease?

Comment by InpharmD Researcher

Per 2022 ICM-VTE guidelines, moderate quality data exists to support tranexamic acid (TXA) use in high-risk orthopedic procedures with prior VTE or other hypercoagulable conditions (e.g., stroke, cancer, atrial fibrillation). Overall, there appears to be a lack of evidence to suggest harm from TXA administration in those with prior VTE history, yet the data are confined to TXA use in limited procedures such as total shoulder arthroplasty or open-heart valvular surgery.

Background

The 2022 International Consensus Group (ICM)-venous thromboembolism (VTE) guidelines provided general recommendations on the risk associated with using tranexamic acid (TXA) and the development of VTE. The panel stated that the administration of TXA in patients undergoing orthopedic procedures does not increase the risk of developing subsequent VTE in patients without prior VTE history (strong recommendation). Even though most patients with prior VTE were excluded in published studies, moderate quality data exists to support TXA use in high-risk orthopedic procedures with prior VTE or other hypercoagulable conditions (e.g., stroke, cancer, atrial fibrillation). A 2017 retrospective matched cohort study of more than 1,200 patients with prior VTE found the risk of recurrent VTE was not significantly greater in patients who received perioperative VTX administration; of the 31 patients who experienced recurrent VTE, TXA administration was not independently associated with increased risk. Another retrospective study of 38,220 total joint arthroplasty patients with prothrombotic conditions also found TXA was not associated with an increase in adverse outcomes in high-risk patients. The decision to utilize TXA must not be solely based on the theoretical risk of VTE, but instead must weigh all risks and benefits to the medication. It is important to note that patients with higher comorbidity burden (e.g., prior VTE, CAD, ASA score ≥ 3, malignancy) are known to have a higher risk of complication following significant blood loss and blood product transfusion and, as such, indirectly benefit from routine TXA usage where there is lack of evidence to suggest harm from TXA administration. [1], [2], [3]

A 2021 retrospective cohort comparison using national claims data (Premier Healthcare) of 71,174 who underwent a total or reverse shoulder arthroplasty identified 9,735 (13.7%) patients in whom the TXA was used during the procedure (34.8% TXA 1,000 mg; 45.8% 2,000 mg TXA). Among TXA users, 1,033 (10.6%) of patients had a history of thrombotic events such as myocardial infarction, DVT, pulmonary embolism, transient ischemic attack, or ischemic stroke (61,439 non-TXA users; 10.5% history of thrombotic events). After adjustment for relevant covariates, overall, TXA use was not associated with increased odds of complications, irrespective of preoperative patient comorbidity burden/risk status. In a subgroup of TXA patients with a history of thrombotic events, TXA use was associated with a slight reduction in hospitalization cost (8.9% CI: 13.1%; 4.6%; p<0.0001; group median $18,830) compared with no TXA use. Based on these findings, the authors concluded among shoulder arthroplasty patients, TXA use was not associated with increased complication odds, independent of a history of thrombotic events. [4]

A 2021 retrospective study investigated the impact of the previous stroke on the risk of TXA-associated seizures. Data were compiled from records of 16,110 patients who had undergone open-heart valvular surgery at a single institution; patients had been given TXA with a bolus of 1 g after heparinization, followed by an infusion of 0.2 g/h until the end of cardiopulmonary bypass. Compared to patients without TXA administration, the adjusted odds ratio (OR) of experiencing a seizure in TXA patients without a history of stroke was 2.44 (95% CI 1.71 to 3.46), whereas in patients receiving TXA with a history of stroke 4.30 (95% CI 2.65 to 6.99). There was no significant interaction between TXA use and preoperative stroke for convulsive seizures. [5]

A 2021 systematic review and meta-analysis examined the association between intravenous TXA with thromboembolic events and mortality. A total of 176 of 219 randomized controlled trials (n= 101 orthopedic studies; n= 6 maxillofacial studies) provided thromboembolic events data (N= 65,900; TXA groups, n= 33,487; Control, n= 32,413). While the incidence of thromboembolic events was higher in the TXA group compared to the control group (2.3% vs. 2.2%), the overall TXA utilization was not significantly associated with an increased risk of thromboembolic events (p= 0.66). Increased risk for vascular occlusive events was not found in studies including patients with a history of thromboembolism. [6]

Additionally, extensive data was available focusing on risk of thrombotic events associated with TXA in general, without focusing specifically on patients with a history of thrombotic events. A 2021 meta-analysis of 234 randomized controlled studies (N= 102,681; 124 in orthopedic surgery) of patients treated with TXA versus no intervention (placebo) found no overall evidence of TXA increasing the risk of thrombotic events (risk ratio [RR] 1.00; 95% CI 0.93 to 1.08; I2= 0%). The risk of VTE, acute coronary syndrome, or stroke was also similar between groups. However, seizures were significantly greater in patients who received more than 2 g/day of TXA (RR 3.05; 95% CI 1.01 to 9.20; p= 0.011). Subgroup analyses based on different types of procedures also did not observe any increase in thrombotic events in trauma (RR 0.89; 95% CI 0.69 to 1.17), obstetrics and gynecology (RR 0.81; 95% CI 0.53 to 1.26), cardiac surgery (RR 0.92; 95% CI 0.81 to 1.05), orthopedic surgery (RR 0.98; 95% CI 0.80 to 1.21). While TXA did not appear to increase the risk of thrombotic events, caution is advised against using higher doses due to the possible increased risk of seizures. [7]

A 2022 meta-analysis investigated the safety and effectiveness of topical TXA in spinal surgery (8 randomized controlled trials, 884 patients). The incidence of VTE was observed in 3.1% (7/226) of the patients in the TXA group and 1.7% (4/229) of patients in the control group (treated with no TXA or isotonic saline). There was no significant difference in the incidence of deep vein thrombosis between the two groups (OR 1.48; 95% CI 0.41 to 5.34, p= 0.55). Based on these findings, the authors suggested that TXA could be safely used during the perioperative period and does not increase the risk of VTE in patients. [8]

Additionally, a 2022 meta-analysis examined the association of TXA administration with mortality and thromboembolic events compared with no treatment or with placebo in patients (aged ≥ 15 years) with traumatic injuries. A total of 31 studies (6 randomized controlled trials and 25 observational studies; N= 43,473) were included for analysis. Due to the significant heterogeneity in regards to 24-hour mortality, a quantitative analysis was not conducted for this outcome. Pooled data for 1-month mortality revealed a significantly decreased mortality in the TXA group compared to the control group (RR 0.83; 95% CI 0.71 to 0.97). Again, substantial heterogeneity was noticed for reported thromboembolic events; estimates of RRs varied from 0.14 (95% CI 0.01 to 2.69) to 24.12 (95% CI 1.42 to 408.88). Thus the risk of VTE remained inconclusive, as 12 studies revealed higher and 8 studies showed lower incidences of thromboembolic events for tranexamic acid treatment compared with the control cohort. [9]

Although TXA has been widely used as a hemostatic adjunct for hemorrhage control in the injured patient, the risk of VTE associated with its use in trauma patients has not been fully evaluated. A 2019 propensity-matched analysis assessed the association between TXA and VTE following trauma in 189 paired patients, with a median Injury Severity Score of 19 and 14 (interquartile range 8-22) in the TXA and non-TXA groups, respectively. The primary outcome of incidence of VTE occurred in 15.3% of patients receiving TXA compared to 7.4% of non-users. Among all VTE events, DVT represented 51.7% and 50.0% of cases in the treated and untreated groups, respectively. The adjusted analysis found TXA to be associated with a significantly higher risk of VTE (adjusted OR [aOR] 3.3; 95% CI 1.3 to 9.1; p= 0.02). The risk of VTE remained elevated in the TXA cohort despite accounting for mortality (subdistribution hazard ratio, 2.42; 95% CI 1.11 to 5.29; p= 0.03). Because the study revealed TXA as an independent risk factor for VTE, the authors suggest carefully selecting injured patients for TXA use is necessary. [10]

References:

[1] ICM-VTE General Delegates. Recommendations from the ICM-VTE: General [published correction appears in J Bone Joint Surg Am. 2022 Aug 3;104(15):e69]. J Bone Joint Surg Am. 2022;104(Suppl 1):4-162. doi:10.2106/JBJS.21.01531
[2] Sabbag OD, Abdel MP, Amundson AW, Larson DR, Pagnano MW. Tranexamic Acid Was Safe in Arthroplasty Patients With a History of Venous Thromboembolism: A Matched Outcome Study. J Arthroplasty. 2017;32(9S):S246-S250. doi:10.1016/j.arth.2017.02.008
[3] Porter SB, White LJ, Osagiede O, Robards CB, Spaulding AC. Tranexamic Acid Administration Is Not Associated With an Increase in Complications in High-Risk Patients Undergoing Primary Total Knee or Total Hip Arthroplasty: A Retrospective Case-Control Study of 38,220 Patients. J Arthroplasty. 2020;35(1):45-51.e3. doi:10.1016/j.arth.2019.08.015
[4] Carbone A, Poeran J, Zubizarreta N, et al. Administration of tranexamic acid during total shoulder arthroplasty is not associated with increased risk of complications in patients with a history of thrombotic events. J Shoulder Elbow Surg. 2021;30(1):104-112. doi:10.1016/j.jse.2020.04.050
[5] Hulde N, Zittermann A, Deutsch MA, von Dossow V, Gummert JF, Koster A. Associations of preoperative stroke and tranexamic acid administration with convulsive seizures in valvular open-heart surgery [published correction appears in J Anesth. 2021 Apr 28;:]. J Anesth. 2021;35(3):451-454. doi:10.1007/s00540-021-02924-w
[6] Taeuber I, Weibel S, Herrmann E, et al. Association of Intravenous Tranexamic Acid With Thromboembolic Events and Mortality: A Systematic Review, Meta-analysis, and Meta-regression [published online ahead of print, 2021 Apr 14]. JAMA Surg. 2021;156(6):e210884. doi:10.1001/jamasurg.2021.0884
[7] Murao S, Nakata H, Roberts I, Yamakawa K. Effect of tranexamic acid on thrombotic events and seizures in bleeding patients: a systematic review and meta-analysis. Crit Care. 2021;25(1):380. Published 2021 Nov 1. doi:10.1186/s13054-021-03799-9
[8] Bao X, Lu H, Gao Z, et al. Meta-Analysis of the Efficacy and Safety of Tranexamic Acid in Spinal Surgery. Comput Math Methods Med. 2022;2022:9406497. Published 2022 Jul 27. doi:10.1155/2022/9406497
[9] Karl V, Thorn S, Mathes T, Hess S, Maegele M. Association of Tranexamic Acid Administration With Mortality and Thromboembolic Events in Patients With Traumatic Injury: A Systematic Review and Meta-analysis. JAMA Netw Open. 2022;5(3):e220625. Published 2022 Mar 1. doi:10.1001/jamanetworkopen.2022.0625
[10] Myers SP, Kutcher ME, Rosengart MR, et al. Tranexamic acid administration is associated with an increased risk of posttraumatic venous thromboembolism. J Trauma Acute Care Surg. 2019;86(1):20-27. doi:10.1097/TA.0000000000002061

Literature Review

A search of the published medical literature revealed 3 studies investigating the researchable question:

Is it safe to use TXA perioperatively in a patient who has a history of stroke, DVT, and sickle cell disease?

Level of evidence

B - One high-quality study or multiple studies with limitations  Read more→



Please see Tables 1-3 for your response.


 

Tranexamic Acid Is Safe in Patients with a History of Coronary Artery Disease Undergoing Total Joint Arthroplasty

Design

Single-center, retrospective study

N= 26,808

Objective

To determine if tranexamic acid (TXA) is safe to use in patients with a history of coronary artery disease (CAD) and cardiovascular stents and to determine if one particular route of administration is safer for these at-risk patients

Study Groups

Patients with or without CAD and stent undergoing TXA/TKA

Inclusion Criteria

Underwent primary total hip arthroplasty (THA) and total knee arthroplasty (TKA)

Exclusion Criteria

Age less than 18 years; underwent nonelective, bilateral, or revision surgery procedure

Methods

Patient data included for analysis were divided into those with a history of CAD or coronary stents which includes any coronary events (e.g., myocardial infarction, pulmonary embolism, deep vein thrombosis) within a 90-day postoperative period. Before September 2017, patients who underwent TKA or THA received 325 mg aspirin PO BID for one month after the operation. After September 2017, only patients at standard risk for VTE have been taking 81 mg aspirin PO BID postoperatively. Anticoagulants such as enoxaparin and rivaroxaban were allowed in select patients with a greater risk of venous thromboembolism (VTE). Any use of previous anticoagulants was kept on regimen through the surgical period.

Patients typically received 2 doses of tranexamic acid (TXA) 1 g IV prior to incision and during would closure. If patients are contraindicated to IV TXA (e.g., history of CAD, recent stents, taking 2 different antiplatelet or anticoagulants), then topical TXA 3 g mixed in 100 mL of saline solution or simply the TXA IV regimen was administered.

Duration

Data collection period: June 2011 to September 2019

Outcome Measures

Primary: Rate of myocardial infarction and VTEs in divided patient groups

Secondary: Difference in outcomes between topical and intravenous TXA in patients undergoing TKA, THA, and total joint arthroplasty (TJA)

Baseline Characteristics

Not reported 

Results

Endpoint

Number of patients

Number of VTEs 

Rate

P-value

Patients with CAD undergoing THA

Patients without CAD undergoing THA

Patients with CAD undergoing TKA

Patients without CAD undergoing TKA

Patients with CAD undergoing THA or TKA

Patients without CAD undergoing THA or TKA

424

12,914

604

12,866

1,028

25,780

1

55

2

141

3

196 

0.235%

0.426%

0.331%

1.096%

0.291%

0.760%

0.560

--

0.073

--

0.086

--

Patients undergoing THA or TKA with coronary stents

Patients undergoing THA or TKA without coronary stents

288

25,780

0

196

0%

0.760%

0.137

--

Stent and topical TXA

Stent and intravenous TXA

162

126

0

0

0%

0%

1

--

TKA procedure

Topical TXA

Intravenous TXA

THA procedure

Topical TXA

Intravenous TXA

TJA procedure

Topical TXA

Intravenous TXA

284

--

--

140

--

--

424

--

--

--

--

--

--

--

--

--

--

--

--

0.546%

0.238%

--

1.053%

0%

--

0.719%

0.133%

0.544

--

--

0.063

--

--

0.123

--

--

Adverse Events

N/A

Study Author Conclusions

In our series, topical and intravenous TXA were equally safe when used in patients with a history of CAD and coronary stents in comparison with the control cohort. With equal efficacy and risk of adverse events, we recommend intravenous TXA, which may enable easier institutional implementation.

InpharmD Researcher Critique

Aside from the risk of selection bias due to the retrospective design, there may have been variability regarding the use of intravenous or topical tranexamic acid as patients with CAD/stents could still receive the intravenous formulation. Anesthesiologists were allowed to practice outside of the institutional protocols based on preference and patient comfort. 



References:

Zak SG, Tang A, Sharan M, Waren D, Rozell JC, Schwarzkopf R. Tranexamic Acid Is Safe in Patients with a History of Coronary Artery Disease Undergoing Total Joint Arthroplasty. J Bone Joint Surg Am. 2021;103(10):900-904. doi:10.2106/JBJS.20.01226

 

Tranexamic acid use and postoperative outcomes in patients undergoing total hip or knee arthroplasty in the United States: retrospective analysis of effectiveness and safety

Design

Multi-center, retrospective cohort study

N= 20,051

Objective

To determine the effectiveness and safety of perioperative tranexamic acid (TXA) use in patients undergoing total hip or knee arthroplasty in the United States

Study Groups

TXA ≤1000 mg (n= 7,041)

TXA= 2000 mg (n= 8,992)

TXA ≥ 3000 mg (n= 4,018)

Inclusion Criteria

Elective total hip or knee arthroplasty

Exclusion Criteria

Unavailable sex information; unknown discharge status; still listed as in-patients at the end of the data collection period; had both a total hip and a total knee arthroplasty during the same hospital stay 

Methods

Utilizing a large national database, this study compared the characteristics and outcomes between patients receiving tranexamic acid and those that did not and analyzed if the use of tranexamic acid is independently associated with altered odds for blood transfusions and perioperative complications, particularly thromboembolic events and acute renal failure. Eligible patients were categorized based on retrieved dosing. 

Duration

January 2006 to October 2012

Outcome Measures

Primary: thromboembolic complications (pulmonary embolism, deep venous thrombosis); combined complications (thromboembolic complications, acute renal failure, cerebrovascular events, myocardial infarction, in-hospital mortality)

Baseline Characteristics

 

Tranexamic acid (n= 20,051)

No tranexamic acid (n= 852,365)

p-value

Age, years

65.9 ± 10.6 65.8 ± 11 0.2554 

Sex

Female

Male

 

12,358 (61.6%)

7,693 (38.4%)

 

518,978 (60.9%)

333,387 (39.1%)

0.0324 

 

 

White

16,578 (82.7%) 645,157 (75.7%)  

Tranexamic acid dose, mg

≤ 1,000

2,000

≥ 3,000

-

7,041 (35.1%) 

8,992 (44.9%)

4,018 (20%)


852,365 (100%)

-

-

-

 

Type of arthroplasty

Unilateral knee

Bilateral knee

Unilateral hip

Bilateral hip

 

12,310 (61.4%)

882 (4.4%)

6,785 (33.8%)

74 (0.4%)

 

545,422 (64%)

34,798 (4.1%)

269,467 (31.6%)

2,678 (0.3%)

<0.001

 

 

 

 

Use of antiplatelet

Aspirin

Other

 

2,602 (13%)

3,591 (17.9%)

 

43,046 (5.1%)

97,608 (11.5%)

 

Use of anticoagulant

Warfarin

Heparin

> 1 or above

 

5,293 (26.4%)

3,142 (15.7%)

5,075 (25.3%)

 

219,407 (25.7%)

225,168 (26.4%)

243,520 (28.6%)

 

Comorbidity

Valvular disease

Pulmonary circulation disease

Peripheral vascular disease

Diabetes

No chronic complications

With chronic complications

Hypertension

Uncomplicated

Complicated

Coagulopathy

 

906 (4.5%)

240 (1.2%)

615 (3.1%)

 

3,703 (18.5%)

335 (1.7%)

 

12,866 (64.2%)

1,055 (5.3%)

848 (4.2%)

 

43,238 (5.1%)

12,010 (1.4%)

26,030 (3.1%)

 

162,615 (19.1%)

15,726 (1.8%)

 

548,962 (64.4%)

44,037 (5.2%)

22,997 (2.7%)

 

0.0004

0.0117

0.9137

 

0.0297

0.0696

 

 0.4863

0.5476

<0.001

Results

Endpoint

TXA ≤1000 mg (n= 7,041)

TXA= 2000 mg (n= 8,992)

TXA ≥ 3000 mg (n= 4,018)

Thromboembolic complications

Odds ratio (95% confidence interval [CI])

 

1.02 (0.71 to 1.45)

 

0.99 (0.70 to 1.39)

 

0.85 (0.53 to 1.35)

Combined complications

Odds ratio (95% CI)

 

0.79 (0.65 to 0.96)*

 

0.75 (0.62 to 0.91)*

 

0.98 (0.78 to 1.24)

* p<0.05

Study Author Conclusions

Tranexamic acid was effective in reducing the need for blood transfusions while not increasing the risk of complications, including thromboembolic events and renal failure. This data provide incremental evidence of the potential effectiveness and safety of tranexamic acid in patients requiring orthopedic surgery.

InpharmD Researcher Critique

Despite multi-center design and the large sample size, this study was limited based on a lack of detailed clinical information (such as hemoglobin levels or other transfusion triggers). Additionally, the study results reported only complications during the hospital stay that may underestimate the actual incidents of complications.



References:

Poeran J, Rasul R, Suzuki S, et al. Tranexamic acid use and postoperative outcomes in patients undergoing total hip or knee arthroplasty in the United States: retrospective analysis of effectiveness and safety. BMJ. 2014;349:g4829. Published 2014 Aug 12. doi:10.1136/bmj.g4829

 

Acute ST-elevation myocardial infarction due to in-stent thrombosis after administering tranexamic acid in a high cardiac risk patient

Design

Case report

Case presentation

A 59-year-old male with a history of total right hip arthroplasty four years prior, known coronary artery disease (CAD), and five drug-eluting coronary stents were admitted for repeat total hip arthroplasty revision due to recurrent prosthetic joint infection. The patient also had hypertension, hyperlipidemia, chronic kidney disease stage II-III, former tobacco use, rare alcohol use, obesity, obstructive sleep apnea, Gilbert's syndrome, and ankylosing spondylitis. Aspirin 81 mg daily was continued and prasugrel was stopped five days prior to the procedure. 

Twenty minutes after the procedure began, tranexamic acid (TXA) was administered as a 500 mg intravenous (IV) bolus dose, followed by another 500 mg IV bolus 10 min later. Three hours after TXA, the ST elevations were identified which could not be confirmed by electrocardiogram (ECG) due to the patient's position. Given the patient's hemodynamic stability, the surgery continued; however, an ECG obtained > 1 hour later found an acute inferolateral STEMI with ST-elevation, and the patient was transferred to the cardiac catheterization laboratory where the patient was successfully treated. Investigations revealed acute in-stent thrombosis with total occlusion in two overlapping stent locations.

Study Author Conclusions

Overlapping stents, bifurcation stents, excessive stent length, and previous in-stent restenosis/thrombosis may increase thrombotic risk. TXA should be administered cautiously with complex stent anatomy.
References:

Kaptein YE. Acute ST-elevation myocardial infarction due to in-stent thrombosis after administering tranexamic acid in a high cardiac risk patient. BMJ Case Rep. 2019;12(4):e227957. Published 2019 Apr 8. doi:10.1136/bcr-2018-227957