Please summarize the efficacy and safety and national guidelines surrounding tafamidis.

Comment by InpharmD Researcher

Tafamidis has demonstrated efficacy in transthyretin amyloid cardiomyopathy (ATTR-CM), with the phase 3 ATTR-ACT trial showing significant reductions in all-cause mortality and cardiovascular-related hospitalizations over 30 months, along with slower decline in functional capacity and quality of life. Safety data indicate adverse event rates comparable to placebo, with no significant treatment-related safety signals. The 2022 AHA/ACC/HFSA guidelines recommend tafamidis for symptomatic (NYHA class I–III) ATTR-CM as the only therapy shown to improve cardiovascular outcomes, and 2024 NICE guidance supports its use within its marketing authorization as a cost-effective option for NHS use. However, high cost and access considerations remain noted limitations.

Background

The 2022 AHA/ACC/HFSA Guideline for the Management of Heart Failure identifies tafamidis as a disease-modifying therapy for transthyretin amyloid cardiomyopathy (ATTR-CM) with demonstrated efficacy in improving cardiovascular outcomes. Specifically, based on the pivotal ATTR-ACT randomized clinical trial, tafamidis significantly reduced all-cause mortality (29.5% vs 42.9%) and cardiovascular-related hospitalizations (0.48 vs 0.70 per year) over 30 months, while also attenuating decline in functional capacity and quality of life. The guideline notes that tafamidis stabilizes transthyretin and prevents further amyloid deposition, with greater benefit when initiated earlier in the disease course, although it does not reverse existing amyloid burden . Safety data indicate that adverse event rates are comparable to placebo, with no significant treatment-related safety signals identified in clinical trials and long-term extension analyses. From a guideline perspective, tafamidis is described as the only therapy shown to improve cardiovascular outcomes in ATTR-CM and is recommended for appropriate patients with symptomatic disease (typically NYHA class I–III), while benefit has not been demonstrated in advanced (class IV) heart failure or certain high-risk populations. Despite its clinical efficacy, the guideline also highlights economic considerations, noting that tafamidis is associated with high cost and low value based on cost-effectiveness analyses. Overall, the guideline supports tafamidis as an evidence-based, outcome-improving therapy for ATTR-CM with a favorable safety profile but acknowledges limitations related to patient selection and cost. [1]

The 2024 NICE technology appraisal guidance recommends tafamidis, within its marketing authorization, as an option for treating wild-type or hereditary ATTR-CM in adults, provided it is supplied under the agreed commercial arrangement. NICE states that ATTR-CM is a progressive, life-limiting condition for which treatment options have largely been limited to symptom management and best supportive care, and identifies tafamidis as the first treatment for ATTR-CM that aims to treat the condition itself. The efficacy evidence considered by the committee was based primarily on the phase 3 ATTR-ACT trial and its open-label long-term extension; NICE reports that the main clinical trial showed tafamidis reduced deaths and hospitalizations from conditions affecting the heart and blood vessels versus placebo, and that longer-term evidence reduced uncertainty regarding survival and treatment duration, although NICE also noted that not all scope-specified updated outcomes, including cardiovascular-related mortality and hospitalizations, were presented at the 84-month follow-up. With respect to safety, NICE notes that ATTR-ACT evaluated the effectiveness, safety, and tolerability of tafamidis versus placebo and that updated adverse event data from the long-term extension were submitted, but the guidance does not report detailed adverse event rates or specific new safety signals in the text provided. From a national guidance perspective, NICE concluded that tafamidis was cost effective versus best supportive care and therefore recommended it for NHS use in England; implementation requirements state that NHS England and integrated care boards should fund access within 30 days of publication because tafamidis had been available through the early access to medicines scheme, and the NHS in Wales must usually provide funding and resources within 2 months of first publication of the final draft guidance. [2]

A 2024 ICER final evidence report on disease-modifying therapies for ATTR-CM states that, in the pivotal ATTR-ACT trial, tafamidis reduced all-cause mortality versus placebo (hazard ratio [HR] 0.67; 95% CI 0.49-0.94), with survival curves diverging at approximately 18 months, reduced cardiovascular-related hospitalizations (0.49 vs 0.70 hospitalizations per year; relative risk ratio 0.70, 95% CI 0.57-0.85), and slowed decline in functional status and quality of life, including a 75.6 m between-group difference in 6-minute walk distance and a 13.4-point difference in KCCQ-OS at 30 months; longer-term follow-up is described as showing a 41% lower risk of all-cause mortality with continuous tafamidis treatment, and ICER judged tafamidis to have high certainty of substantial net health benefit in the original trial population and, in a contemporary population, high certainty of at least small net health benefit with moderate certainty of substantial net health benefit. Safety was described as favorable and comparable to placebo and to the 20 mg dose, with most adverse events mild or moderate; the most common adverse events were diarrhea (8%) in the 80 mg group and urinary tract infection (5.7%) in the 20 mg group, and dose reductions were uncommon (1.1% with tafamidis 80 mg vs 2.3% with placebo). Regarding guidelines, the report summarizes that the 2023 World Heart Federation consensus notes strong evidence from ATTR-ACT supporting tafamidis and highlights access and cost barriers; the 2023 ACC Expert Consensus Decision Pathway describes tafamidis as effective with a favorable side-effect profile but identifies cost and copayment-navigation barriers; the 2022 AHA/ACC/HFSA heart failure guideline recommends tafamidis for select patients with wild-type or hereditary ATTR-CM and NYHA class I-III symptoms to reduce cardiovascular morbidity and mortality (Class 1, Level B); and the 2020 Canadian Cardiovascular Society/Canadian Heart Failure Society position statement notes the efficacy of tafamidis in ATTR-ACT and states that treatment choice in patients with mixed cardiac and neurologic phenotypes should be individualized by interdisciplinary teams. [3]

These phase 3 ATTR-ACT and long-term extension (LTE) analyses in transthyretin amyloid cardiomyopathy report that tafamidis was associated with reductions in mortality, cardiovascular-related hospitalizations, functional decline, and biomarker progression, with a safety profile described as comparable to placebo. In ATTR-ACT, tafamidis 80 mg and 20 mg both significantly reduced the composite of all-cause mortality and cardiovascular-related hospitalizations versus placebo (p= 0.0030 and p= 0.0048, respectively), reduced decline in 6-minute walk test distance and KCCQ-OS scores (p<0.0001 for both doses), and lowered rates of cardiovascular-related hospitalizations; all-cause mortality was significantly reduced with 80 mg (hazard ratio [HR] 0.69; 95% CI 0.487 to 0.979; p= 0.0378), while 20 mg showed a non-significant reduction (HR 0.715; p= 0.1564). Tafamidis 80 mg also demonstrated greater attenuation of increases in NT-proBNP and troponin I compared with placebo, with a significant difference versus 20 mg for NT-proBNP. Long-term data showed that patients initially treated with tafamidis had lower all-cause mortality than those initially receiving placebo and later transitioning to tafamidis (HR 0.59; 95% CI 0.44 to 0.79; p<0.001) over a median follow-up of approximately 58 months, with consistent effects across genotype and NYHA class subgroups. Across studies, tafamidis was reported as generally well tolerated, with similar rates of adverse events, serious adverse events, and discontinuations compared with placebo, and no new safety concerns identified in the LTE. [4], [5]

References: [1] Heidenreich PA, Bozkurt B, Aguilar D, et al. 2022 AHA/ACC/HFSA guideline for the management of heart failure: a report of the American College of Cardiology/American Heart Association Joint Committee on Clinical Practice Guidelines. Circulation. 2022;145:e895–e1032. doi:10.1161/CIR.0000000000001063
[2] National Institute for Health and Care Excellence (NICE). Tafamidis for treating transthyretin amyloidosis with cardiomyopathy (TA984). Published June 19, 2024. Accessed 2026.
[3] Wasfy JH, Winn AN, Touchette DR, Nikitin D, Shah KK, Richardson M, Lee W, Kim S, Rind DM. Disease modifying therapies for the treatment of transthyretin amyloid cardiomyopathy (ATTR-CM): final evidence report. Institute for Clinical and Economic Review; October 21, 2024.
[4] Elliott P, Drachman BM, Gottlieb SS, et al. Long-Term Survival With Tafamidis in Patients With Transthyretin Amyloid Cardiomyopathy. Circ Heart Fail. 2022;15(1):e008193. doi:10.1161/CIRCHEARTFAILURE.120.008193
[5] Damy T, Garcia-Pavia P, Hanna M, et al. Efficacy and safety of tafamidis doses in the Tafamidis in Transthyretin Cardiomyopathy Clinical Trial (ATTR-ACT) and long-term extension study. Eur J Heart Fail. 2021;23(2):277-285. doi:10.1002/ejhf.2027
Literature Review

A search of the published medical literature revealed 1 study investigating the researchable question:

Please summarize the efficacy and safety and national guidelines surrounding tafamidis.

Level of evidence

B - One high-quality study or multiple studies with limitations  Read more→



Please see Table 1 for your response.


Tafamidis Treatment for Patients with Transthyretin Amyloid Cardiomyopathy

Design

Multicenter, international, double-blind, placebo-controlled, phase 3 trial

N= 441

Objective

To assess the efficacy and safety of tafamidis in reducing all-cause mortality and cardiovascular-related hospitalizations in patients with transthyretin amyloid cardiomyopathy

Study Groups

Tafamidis 80 mg (n= 176)

Tafamidis 20 mg (n= 88)

Placebo (n= 177)

Inclusion Criteria

Patients aged 18-90 with transthyretin amyloid cardiomyopathy confirmed by amyloid deposits on biopsy and transthyretin precursor protein confirmed by immunohistochemical analysis, scintigraphy, or mass spectrometry; cardiac involvement confirmed by echocardiography and history of heart failure

Exclusion Criteria

Heart failure not due to transthyretin amyloid cardiomyopathy, NYHA class IV heart failure, light-chain amyloidosis, history of liver or heart transplantation, implanted cardiac device, previous tafamidis treatment, eGFR <25 ml/min/1.73 m2, liver transaminase levels >2x upper limit of normal, severe malnutrition, concurrent treatment with NSAIDs, tauroursodeoxycholate, doxycycline, calcium-channel blockers, or digitalis

Methods

Patients were randomly assigned to receive 80 mg or 20 mg of tafamidis or placebo daily for 30 months. The primary analysis assessed all-cause mortality and cardiovascular-related hospitalizations using the Finkelstein–Schoenfeld method. Secondary endpoints included changes in the 6-minute walk test and KCCQ-OS score. Safety was monitored throughout the trial.

Duration

30 months

Outcome Measures

Primary: All-cause mortality, cardiovascular-related hospitalizations

Secondary: Change in 6-minute walk test distance, change in KCCQ-OS score

Baseline Characteristics  

Tafamidis (N= 264)

Placebo (N= 177)
Age, mean years

74.5 ± 7.2

74.1 ± 6.7
Male

241 (91.3%)

157 (88.7%)
ATTRm

63 (23.9%)

43 (24.3%)
ATTRwt

201 (76.1%)

134 (75.7%)
NYHA Class I

24 (9.1%)

13 (7.3%)
NYHA Class II

162 (61.4%)

101 (57.1%)
NYHA Class III

78 (29.5%)

63 (35.6%)
Results  

Tafamidis (N= 264)

Placebo (N= 177) p-value
All-cause mortality

78 (29.5%)

76 (42.9%) <0.001
Cardiovascular-related hospitalizations per year

0.48

0.70 <0.001
6-minute walk test change (m)

-75.68

- <0.001
KCCQ-OS score change

-13.65

- <0.001
Adverse Events

The incidence and types of adverse events were similar in the tafamidis and placebo groups. Common adverse events included diarrhea and urinary tract infections, which were less common in the tafamidis group. Permanent discontinuation due to adverse events was less common in the tafamidis group.

Study Author Conclusions

In patients with transthyretin amyloid cardiomyopathy, tafamidis was associated with reductions in all-cause mortality and cardiovascular-related hospitalizations and reduced the decline in functional capacity and quality of life as compared with placebo.

Critique

The study's strengths include its large sample size and rigorous design. However, the trial's exclusion criteria may limit the generalizability of the findings to all patients with transthyretin amyloid cardiomyopathy. Additionally, the study did not explore the long-term effects beyond 30 months.

 

References:
[1] [1] Maurer MS, Schwartz JH, Gundapaneni B, et al; ATTR-ACT Study Investigators. Tafamidis treatment for patients with transthyretin amyloid cardiomyopathy. N Engl J Med. 2018;379(11):1007-1016. doi:10.1056/NEJMoa1805689